For: | Broekman F, Giovannetti E, Peters GJ. Tyrosine kinase inhibitors: Multi-targeted or single-targeted? World J Clin Oncol 2011; 2(2): 80-93 [PMID: 21603317 DOI: 10.5306/wjco.v2.i2.80] |
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URL: | https://www.wjgnet.com/2218-4333/full/v2/i2/80.htm |
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Aishwarya Shinde, Kanan Panchal, Sumeet Katke, Rishi Paliwal, Akash Chaurasiya. Tyrosine kinase inhibitors as next generation oncological therapeutics: Current strategies, limitations and future perspectives. Therapies 2022; 77(4): 425 doi: 10.1016/j.therap.2021.10.010
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Aleksandra Sochacka-Ćwikła, Marcin Mączyński, Andrzej Regiec. FDA-Approved Small Molecule Compounds as Drugs for Solid Cancers from Early 2011 to the End of 2021. Molecules 2022; 27(7): 2259 doi: 10.3390/molecules27072259
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Maria Kalyukina, Yuliana Yosaatmadja, Martin J. Middleditch, Adam V. Patterson, Jeff B. Smaill, Christopher J. Squire. TAS‐120 Cancer Target Binding: Defining Reactivity and Revealing the First Fibroblast Growth Factor Receptor 1 (FGFR1) Irreversible Structure. ChemMedChem 2019; 14(4): 494 doi: 10.1002/cmdc.201800719
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Models of Nanostructures Based on Titanium Dioxide TiO for Transport of Biologically Active Compounds. Nanosistemi, Nanomateriali, Nanotehnologii 2020; 18(4) doi: 10.15407/nnn.18.04.1077
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Areej Abuhammad, Mutasem Taha. Innovative Computer-Aided Methods for the Discovery of New Kinase Ligands. Future Medicinal Chemistry 2016; 8(5): 509 doi: 10.4155/fmc-2015-0003
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Sanja Aveic, Gian Paolo Tonini. Resistance to receptor tyrosine kinase inhibitors in solid tumors: can we improve the cancer fighting strategy by blocking autophagy?. Cancer Cell International 2016; 16(1) doi: 10.1186/s12935-016-0341-2
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Mingyue Luo, Lu Sun, Rongping Dai, Youxin Chen, Chan Wu. Central retinal vein occlusion in patients with metastatic solid tumors on tyrosine kinase inhibitors: a report of case series and literature review. Frontiers in Medicine 2024; 11 doi: 10.3389/fmed.2024.1362108
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Cristina Olgasi, Patrizia Dentelli, Arturo Rosso, Alessandra Iavello, Gabriele Togliatto, Valentina Toto, Marcella Liberatore, Giuseppina Barutello, Piero Musiani, Federica Cavallo, Maria Felice Brizzi. DNA vaccination against membrane-bound Kit ligand: A new approach to inhibiting tumour growth and angiogenesis. European Journal of Cancer 2014; 50(1): 234 doi: 10.1016/j.ejca.2013.09.016
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Eman A. Abd El-Meguid, Ahmed M. Naglah, Gaber O. Moustafa, Hanem M. Awad, Ahmed M. El Kerdawy. Novel benzothiazole-based dual VEGFR-2/EGFR inhibitors targeting breast and liver cancers: Synthesis, cytotoxic activity, QSAR and molecular docking studies. Bioorganic & Medicinal Chemistry Letters 2022; 58: 128529 doi: 10.1016/j.bmcl.2022.128529
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10 |
Darawan Rinchai, Elena Verzoni, Veronica Huber, Agata Cova, Paola Squarcina, Loris De Cecco, Filippo de Braud, Raffaele Ratta, Matteo Dugo, Luca Lalli, Viviana Vallacchi, Monica Rodolfo, Jessica Roelands, Chiara Castelli, Damien Chaussabel, Giuseppe Procopio, Davide Bedognetti, Licia Rivoltini. Integrated transcriptional‐phenotypic analysis captures systemic immunomodulation following antiangiogenic therapy in renal cell carcinoma patients. Clinical and Translational Medicine 2021; 11(6) doi: 10.1002/ctm2.434
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11 |
Xiaoxiao Sun, Qiaoling Song, Li He, Lei Yan, Jingli Liu, Qing Zhang, Qiang Yu. Receptor Tyrosine Kinase Phosphorylation Pattern–Based Multidrug Combination Is an Effective Approach for Personalized Cancer Treatment. Molecular Cancer Therapeutics 2016; 15(10): 2508 doi: 10.1158/1535-7163.MCT-15-0735
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12 |
Simone De Leo, Matteo Trevisan, Claudia Moneta, Carla Colombo. Endocrine-related adverse conditions induced by tyrosine kinase inhibitors. Annales d'Endocrinologie 2023; 84(3): 374 doi: 10.1016/j.ando.2023.03.009
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13 |
Giuseppe Tridente. Adverse Events and Oncotargeted Kinase Inhibitors. 2017; : 695 doi: 10.1016/B978-0-12-809400-6.00029-9
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14 |
Sareshma Sudhesh Dev, Syafiq Asnawi Zainal Abidin, Reyhaneh Farghadani, Iekhsan Othman, Rakesh Naidu. Receptor Tyrosine Kinases and Their Signaling Pathways as Therapeutic Targets of Curcumin in Cancer. Frontiers in Pharmacology 2021; 12 doi: 10.3389/fphar.2021.772510
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Jijin Wang, Di Huang, Wenjing Yang, Qingxu Song, Yibin Jia, Pengxiang Chen, Yufeng Cheng. The efficacy and safety of Apatinib in the treatment of advanced non-small cell lung cancer: A retrospective trial. Frontiers in Oncology 2022; 12 doi: 10.3389/fonc.2022.1030798
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16 |
Bashdar Mahmud Hussen, Khozga Hazhar Abdullah, Snur Rasool Abdullah, Nasik Mahmood Majeed, Sayran Mohamadtahr, Mohammed Fatih Rasul, Peixin Dong, Mohammad Taheri, Majid Samsami. New insights of miRNA molecular mechanisms in breast cancer brain metastasis and therapeutic targets. Non-coding RNA Research 2023; 8(4): 645 doi: 10.1016/j.ncrna.2023.09.003
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17 |
Priyanka Gupta, Keehn Strange, Rahul Telange, Ailan Guo, Heather Hatch, Amin Sobh, Jonathan Elie, Angela M. Carter, John Totenhagen, Chunfeng Tan, Yogesh A. Sonawane, Jiri Neuzil, Amarnath Natarajan, Ashley J. Ovens, Jonathan S. Oakhill, Thorsten Wiederhold, Karel Pacak, Hans K. Ghayee, Laurent Meijer, Sushanth Reddy, James Bibb. Genetic Impairment of Succinate Metabolism Disrupts Bioenergetic Sensing in Adrenal Neuroendocrine Cancer. SSRN Electronic Journal 2022; doi: 10.2139/ssrn.4018612
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18 |
Venice Wing Tung Ho, Hor Yue Tan, Ning Wang, Yibin Feng. Tyrosine Kinases as Druggable Targets in Cancer. 2019; doi: 10.5772/intechopen.82513
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19 |
Charles Pottier, Margaux Fresnais, Marie Gilon, Guy Jérusalem, Rémi Longuespée, Nor Eddine Sounni. Tyrosine Kinase Inhibitors in Cancer: Breakthrough and Challenges of Targeted Therapy. Cancers 2020; 12(3): 731 doi: 10.3390/cancers12030731
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20 |
Maša Kenda, Damjan Avsec, Taja Zore, Eva Kogovšek, Urša Pečar Fonović, Janko Kos, Krištof Bozovičar, Tomaž Bratkovič, Nataša Karas Kuželički, Bojana Žegura, Metka Filipič, Marija Sollner Dolenc. Effects of tyrosine kinase inhibitors on androgen, estrogen α, glucocorticoid and thyroid receptors. Toxicology and Applied Pharmacology 2022; 434: 115818 doi: 10.1016/j.taap.2021.115818
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Siva M Gangadhar, Mithilesh Yadav, Nishith S Mandal. Dermatofibrosarcoma Protuberans: A Surgeon's Enigma. Cureus 2023; doi: 10.7759/cureus.44144
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22 |
Mustafa A. Al-Qadhi, Heba Abdelrasheed Allam, Samar H. Fahim, Tawfeek A.A. Yahya, Fatma A.F. Ragab. Design and synthesis of certain 7-Aryl-2-Methyl-3-Substituted Pyrazolo{1,5-a}Pyrimidines as multikinase inhibitors. European Journal of Medicinal Chemistry 2023; 262: 115918 doi: 10.1016/j.ejmech.2023.115918
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23 |
Jian Wu, Suresh Kumar, Feng Wang, Hui Wang, Lijia Chen, Patrick Arsenault, Michael Mattern, Joseph Weinstock. Chemical Approaches to Intervening in Ubiquitin Specific Protease 7 (USP7) Function for Oncology and Immune Oncology Therapies. Journal of Medicinal Chemistry 2018; 61(2): 422 doi: 10.1021/acs.jmedchem.7b00498
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Francesco Sabbatino, Valeria Conti, Luigi Liguori, Giovanna Polcaro, Graziamaria Corbi, Valentina Manzo, Vincenzo Tortora, Chiara Carlomagno, Carmine Vecchione, Amelia Filippelli, Stefano Pepe. Molecules and Mechanisms to Overcome Oxidative Stress Inducing Cardiovascular Disease in Cancer Patients. Life 2021; 11(2): 105 doi: 10.3390/life11020105
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Aiten M. Soliman, Mostafa M. Ghorab. Exploration of N-alkyl-2-[(4-oxo-3-(4-sulfamoylphenyl)-3,4-dihydroquinazolin-2-yl)thio]acetamide derivatives as anticancer and radiosensitizing agents. Bioorganic Chemistry 2019; 88: 102956 doi: 10.1016/j.bioorg.2019.102956
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Anh Thu Vu, Lara Akingunsade, Konstantin Hoffer, Cordula Petersen, Christian Stephan Betz, Kai Rothkamm, Thorsten Rieckmann, Lara Bussmann, Malte Kriegs. Src family kinase targeting in head and neck tumor cells using SU6656, PP2 and dasatinib. Head & Neck 2023; 45(1): 147 doi: 10.1002/hed.27216
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Eman M.E. Dokla, Amal Kamal Abdel-Aziz, Sandra N. Milik, Amr H. Mahmoud, Mona Kamal Saadeldin, Martin J. McPhillie, Saverio Minucci, Khaled A.M. Abouzid. Indolin-2-one derivatives as selective Aurora B kinase inhibitors targeting breast cancer. Bioorganic Chemistry 2021; 117: 105451 doi: 10.1016/j.bioorg.2021.105451
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28 |
Robert I. Haddad, Martin Schlumberger, Lori J. Wirth, Eric J. Sherman, Manisha H. Shah, Bruce Robinson, Corina E. Dutcus, Angela Teng, Andrew G. Gianoukakis, Steven I. Sherman. Incidence and timing of common adverse events in Lenvatinib-treated patients from the SELECT trial and their association with survival outcomes. Endocrine 2017; 56(1): 121 doi: 10.1007/s12020-017-1233-5
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Shelly Pathania, Olli T. Pentikäinen, Pankaj Kumar Singh. A holistic view on c-Kit in cancer: Structure, signaling, pathophysiology and its inhibitors. Biochimica et Biophysica Acta (BBA) - Reviews on Cancer 2021; 1876(2): 188631 doi: 10.1016/j.bbcan.2021.188631
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Bibian M. E. Tullemans, Magdolna Nagy, Siamack Sabrkhany, Arjan W. Griffioen, Mirjam G. A. oude Egbrink, Maureen Aarts, Johan W. M. Heemskerk, Marijke J. E. Kuijpers. Tyrosine Kinase Inhibitor Pazopanib Inhibits Platelet Procoagulant Activity in Renal Cell Carcinoma Patients. Frontiers in Cardiovascular Medicine 2018; 5 doi: 10.3389/fcvm.2018.00142
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31 |
Sanjay K. Srikakulam, Tomas Bastys, Olga V. Kalinina. A shift of dynamic equilibrium between the KIT active and inactive states causes drug resistance. Proteins: Structure, Function, and Bioinformatics 2020; 88(11): 1434 doi: 10.1002/prot.25963
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Samy Mohamady, Mahmoud Galal, Wagdy M. Eldehna, David C. Gutierrez, Hany S. Ibrahim, Mohey M. Elmazar, Hamed I. Ali. Dual Targeting of VEGFR2 and C-Met Kinases via the Design and Synthesis of Substituted 3-(Triazolo-thiadiazin-3-yl)indolin-2-one Derivatives as Angiogenesis Inhibitors. ACS Omega 2020; 5(30): 18872 doi: 10.1021/acsomega.0c02038
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Adriana Zámečníkova. Novel approaches to the development of tyrosine kinase inhibitors and their role in the fight against cancer. Expert Opinion on Drug Discovery 2014; 9(1): 77 doi: 10.1517/17460441.2014.865012
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E. A. Shatokhina, L. S. Kruglova, A. S. Polonskaia. Management of acneiform rash associated with anti-EGFR monoclonal antibody treatment. Meditsinskiy sovet = Medical Council 2020; (20): 157 doi: 10.21518/2079-701X-2020-20-157-164
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35 |
Nurmaya Effendi, Kenji Mishiro, Takeshi Takarada, Akira Makino, Daisuke Yamada, Yoji Kitamura, Kazuhiro Shiba, Yasushi Kiyono, Akira Odani, Kazuma Ogawa. Radiobrominated benzimidazole-quinoline derivatives as Platelet-derived growth factor receptor beta (PDGFRβ) imaging probes. Scientific Reports 2018; 8(1) doi: 10.1038/s41598-018-28529-0
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36 |
Wen-Hsing Lin, Su-Ying Wu, Teng-Kuang Yeh, Chiung-Tong Chen, Jen-Shin Song, Hui-Yi Shiao, Ching-Chuan Kuo, Tsu Hsu, Cheng-Tai Lu, Pei-Chen Wang, Tsung-Sheng Wu, Yi-Hui Peng, Hui-You Lin, Ching-Ping Chen, Ya-Ling Weng, Fang-Chun Kung, Mine-Hsine Wu, Yu-Chieh Su, Kuo-Wei Huang, Ling-Hui Chou, Ching-Cheng Hsueh, Kuei-Jung Yen, Po-Chu Kuo, Chen-Lung Huang, Li-Tzong Chen, Chuan Shih, Hui-Jen Tsai, Weir-Torn Jiaang. Identification of a Multitargeted Tyrosine Kinase Inhibitor for the Treatment of Gastrointestinal Stromal Tumors and Acute Myeloid Leukemia. Journal of Medicinal Chemistry 2019; 62(24): 11135 doi: 10.1021/acs.jmedchem.9b01229
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37 |
Wagdy M. Eldehna, Ahmed M. El Kerdawy, Ghada H. Al-Ansary, Sara T. Al-Rashood, Mamdouh M. Ali, Abeer E. Mahmoud. Type IIA - Type IIB protein tyrosine kinase inhibitors hybridization as an efficient approach for potent multikinase inhibitor development: Design, synthesis, anti-proliferative activity, multikinase inhibitory activity and molecular modeling of novel indolinone-based ureides and amides. European Journal of Medicinal Chemistry 2019; 163: 37 doi: 10.1016/j.ejmech.2018.11.061
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38 |
Kyaw Zwar Myint, Brinda Balasubramanian, Simran Venkatraman, Suchada Phimsen, Supisara Sripramote, Jeranan Jantra, Chaiwat Choeiphuk, Somkit Mingphruedhi, Paramin Muangkaew, Narongsak Rungsakulkij, Pongsatorn Tangtawee, Wikran Suragul, Watoo Vassanasiri Farquharson, Kanokpan Wongprasert, Somchai Chutipongtanate, Pimtip Sanvarinda, Marisa Ponpuak, Naravat Poungvarin, Tavan Janvilisri, Tuangporn Suthiphongchai, Kiren Yacqub-Usman, Anna M. Grabowska, David O. Bates, Rutaiwan Tohtong. Therapeutic Implications of Ceritinib in Cholangiocarcinoma beyond ALK Expression and Mutation. Pharmaceuticals 2024; 17(2): 197 doi: 10.3390/ph17020197
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39 |
Giuseppe Tridente. Adverse Events and Oncotargeted Kinase Inhibitors. 2017; : 145 doi: 10.1016/B978-0-12-809400-6.00007-X
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40 |
Josep Tabernero, Rocio Garcia-Carbonero, James Cassidy, Alberto Sobrero, Eric Van Cutsem, Claus-Henning Köhne, Sabine Tejpar, Oleg Gladkov, Irina Davidenko, Ramon Salazar, Liubov Vladimirova, Sergey Cheporov, Olga Burdaeva, Fernando Rivera, Leslie Samuel, Irina Bulavina, Vanessa Potter, Yu-Lin Chang, Nathalie A. Lokker, Peter J. O'Dwyer. Sorafenib in Combination with Oxaliplatin, Leucovorin, and Fluorouracil (Modified FOLFOX6) as First-line Treatment of Metastatic Colorectal Cancer: The RESPECT Trial. Clinical Cancer Research 2013; 19(9): 2541 doi: 10.1158/1078-0432.CCR-13-0107
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Wenjing Xu, Chunping Ye, Xin Qing, Shengli Liu, Xinyi Lv, Wenjun Wang, Xiaochen Dong, Yewei Zhang. Multi-target tyrosine kinase inhibitor nanoparticle delivery systems for cancer therapy. Materials Today Bio 2022; 16: 100358 doi: 10.1016/j.mtbio.2022.100358
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Valentina Gandin, Alessandro Ferrarese, Martina Dalla Via, Cristina Marzano, Adriana Chilin, Giovanni Marzaro. Targeting kinases with anilinopyrimidines: discovery of N-phenyl-N’-[4-(pyrimidin-4-ylamino)phenyl]urea derivatives as selective inhibitors of class III receptor tyrosine kinase subfamily. Scientific Reports 2015; 5(1) doi: 10.1038/srep16750
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Fares Hezam Al-Ostoot, Ankith Sherapura, Vikas H. Malojirao, Prabhu Thirusangu, Tahani I. Al-Muhimeed, Shaukath Ara Khanum, B. T. Prabhakar. Modulation of DNA damage response by targeting ATM kinase using newly synthesized di-phenoxy acetamide (DPA) analogs to induce anti-neoplasia. Pharmacological Reports 2021; 73(5): 1344 doi: 10.1007/s43440-021-00292-6
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Gabor Valcz, Ferenc Sipos, Zsolt Tulassay, Bela Molnar, Yukako Yagi. Republished: Importance of carcinoma-associated fibroblast-derived proteins in clinical oncology. Postgraduate Medical Journal 2015; 91(1075): 291 doi: 10.1136/postgradmedj-2014-202561rep
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Rania Kheder El-Fekih, Clément Deltombe, Hassan Izzedine. Microangiopathie thrombotique et cancer. Néphrologie & Thérapeutique 2017; 13(6): 439 doi: 10.1016/j.nephro.2017.01.023
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Sheetal Chauhan, Seema Sen, Khushboo Irshad, Seema Kashyap, Neelam Pushker, Rachna Meel, Mehar Chand Sharma. Receptor tyrosine kinase gene expression profiling of orbital rhabdomyosarcoma unveils MET as a potential biomarker and therapeutic target. Human Cell 2023; 37(1): 297 doi: 10.1007/s13577-023-00993-5
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Sindhu M. Parameshwaraiah, Rashmi Shivakumar, Zhang Xi, Tejaswini P. Siddappa, Akshay Ravish, Arunkumar Mohan, Lisha K. Poonacha, Pradeep M. Uppar, Shreeja Basappa, Dukanya Dukanya, Santhosh L. Gaonkar, Kempaiah Kemparaju, Peter E. Lobie, Vijay Pandey, Basappa Basappa. Development of Novel Indazolyl‐Acyl Hydrazones as Antioxidant and Anticancer Agents that Target VEGFR‐2 in Human Breast Cancer Cells. Chemistry & Biodiversity 2024; 21(3) doi: 10.1002/cbdv.202301950
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Megan L. Troxell, John P. Higgins, Neeraja Kambham. Antineoplastic Treatment and Renal Injury: An Update on Renal Pathology Due to Cytotoxic and Targeted Therapies. Advances in Anatomic Pathology 2016; 23(5): 310 doi: 10.1097/PAP.0000000000000122
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Zachary S. Peacock, Deepak Kademani, Anh D. Le, Janice S. Lee, Robert G. Hale, Larry L. Cunningham. Proceedings From the 2011 American Association of Oral and Maxillofacial Surgeons Research Summit. Journal of Oral and Maxillofacial Surgery 2012; 70(6): 1271 doi: 10.1016/j.joms.2012.01.029
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Josep Esteve Romero, Jaume Albiol Chiva, Juan Peris-Vicente, Enrique Ochoa-Aranda. Development and Validation of A Micellar Liquid Chromatographic Method to Determine Three Antitumorals in Plasma. Bioanalysis 2017; 9(10): 799 doi: 10.4155/bio-2017-0028
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Aliaksandr Faryna, Elena Kalinichenko. Molecular Docking - Recent Advances. Biomedical Engineering 2023; 15 doi: 10.5772/intechopen.107236
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Amirrtha Srikanthan, Josee-Lyne Ethier, Alberto Ocana, Bostjan Seruga, Monika K. Krzyzanowska, Eitan Amir, Jung Weon Lee. Cardiovascular Toxicity of Multi-Tyrosine Kinase Inhibitors in Advanced Solid Tumors: A Population-Based Observational Study. PLOS ONE 2015; 10(3): e0122735 doi: 10.1371/journal.pone.0122735
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Jianbiao Zhou, Wee-Joo Chng. Resistance to FLT3 inhibitors in acute myeloid leukemia: Molecular mechanisms and resensitizing strategies. World Journal of Clinical Oncology 2018; 9(5): 90-97 doi: 10.5306/wjco.v9.i5.90
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Gabor Valcz, Ferenc Sipos, Zsolt Tulassay, Bela Molnar, Yukako Yagi. Importance of carcinoma-associated fibroblast-derived proteins in clinical oncology. Journal of Clinical Pathology 2014; 67(12): 1026 doi: 10.1136/jclinpath-2014-202561
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Mohammed S. Abdel-Maksoud, Hebatollah E. Eitah, Rasha M. Hassan, Walaa Hamada Abd-Allah. Design and synthesis of novel pyrimidine-pyrazole hybrids with dual anticancer and anti-inflammatory effects targeting BRAFV600E and JNK. Molecular Diversity 2025; doi: 10.1007/s11030-025-11121-w
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Haoyue Guo, Binglei Li, Li Diao, Hao Wang, Peixin Chen, Minlin Jiang, Lishu Zhao, Yayi He, Caicun Zhou. An immune-based risk-stratification system for predicting prognosis in pulmonary sarcomatoid carcinoma (PSC). OncoImmunology 2021; 10(1) doi: 10.1080/2162402X.2021.1947665
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Krisyanti Budipramana, Frangky Sangande. Structural and molecular insights from dual inhibitors of EGFR and VEGFR2 as a strategy to improve the efficacy of cancer therapy. Chemical Biology & Drug Design 2024; 103(5) doi: 10.1111/cbdd.14534
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Giuseppe Tridente. Adverse Events and Oncotargeted Kinase Inhibitors. 2017; : 57 doi: 10.1016/B978-0-12-809400-6.00003-2
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Anna M. Ogloblina, Alexandra N. Khristich, Natalia Y. Karpechenko, Svetlana E. Semina, Gennady A. Belitsky, Nina G. Dolinnaya, Marianna G. Yakubovskaya. Multi-targeted effects of G4-aptamers and their antiproliferative activity against cancer cells. Biochimie 2018; 145: 163 doi: 10.1016/j.biochi.2017.11.020
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Aik-Choon Tan, Simon Vyse, Paul H. Huang. Exploiting receptor tyrosine kinase co-activation for cancer therapy. Drug Discovery Today 2017; 22(1): 72 doi: 10.1016/j.drudis.2016.07.010
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Katie Bechman, James B Galloway, Kevin L Winthrop. Small-Molecule Protein Kinases Inhibitors and the Risk of Fungal Infections. Current Fungal Infection Reports 2019; 13(4): 229 doi: 10.1007/s12281-019-00350-w
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Elizabeth Irvine, Casey Williams. Treatment-, Patient-, and Disease-Related Factors and the Emergence of Adverse Events with Tyrosine Kinase Inhibitors for the Treatment of Chronic Myeloid Leukemia. Pharmacotherapy: The Journal of Human Pharmacology and Drug Therapy 2013; 33(8): 868 doi: 10.1002/phar.1266
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Mike-Andrew Westhoff, Nicolas Marschall, Klaus-Michael Debatin. Apoptosis in Cancer Pathogenesis and Anti-cancer Therapy. Advances in Experimental Medicine and Biology 2016; 930: 173 doi: 10.1007/978-3-319-39406-0_8
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Kadri Valter, Boris Zhivotovsky, Vladimir Gogvadze. Cell death-based treatment of neuroblastoma. Cell Death & Disease 2018; 9(2) doi: 10.1038/s41419-017-0060-1
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Nadia Panera, Annalisa Crudele, Ilaria Romito, Daniela Gnani, Anna Alisi. Focal Adhesion Kinase: Insight into Molecular Roles and Functions in Hepatocellular Carcinoma. International Journal of Molecular Sciences 2017; 18(1): 99 doi: 10.3390/ijms18010099
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Mohamed Mokhtar, Khadijah S. Alghamdi, Nesreen S. Ahmed, Dina Bakhotmah, Tamer S. Saleh. Design and green synthesis of novel quinolinone derivatives of potential anti-breast cancer activity against MCF-7 cell line targeting multi-receptor tyrosine kinases. Journal of Enzyme Inhibition and Medicinal Chemistry 2021; 36(1): 1453 doi: 10.1080/14756366.2021.1944126
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Maninder Kaur, Pankaj Kumar Singh, Manjinder Singh, Renu Bahadur, Om Silakari. Molecular dynamics and integrated pharmacophore-based identification of dual $$\hbox {JAK3/PI3K}\delta $$ JAK3/PI3K δ inhibitors. Molecular Diversity 2018; 22(1): 95 doi: 10.1007/s11030-017-9794-z
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Halyna M. Kuznietsova, Vasyl V. Hurmach, Andriy V. Bychko, Olena I. Tykhoniuk, Demyd S. Milokhov, Olga V. Khilya, Yulian M. Volovenko, Volodymyr K. Rybalchenko. Synthesis and biological activity of 4-amino-3-chloro-1H-pyrrole-2,5-diones. In Silico Pharmacology 2019; 7(1) doi: 10.1007/s40203-019-0051-2
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Wagdy M. Eldehna, Eslam Roshdy, Maha-Hamadien Abdulla, Abdelrahman I. Zain-Alabdeen, Moataz A. Shaldam, Noura S. Alhassan, Thamer Bin Traiki, Mohammad M. Al-Sanea, Anwar A. El-Hamaky, Ahmed A. Al-Karmalawy, Ahmed M. El Kerdawy, Manabu Abe, Haytham O. Tawfik. Discovery of 1-phenyl-1,2,3-triazole ureas as dual VEGFR-2/JNK-1 type II kinase inhibitors targeting pancreatic cancer. International Journal of Biological Macromolecules 2025; 308: 142372 doi: 10.1016/j.ijbiomac.2025.142372
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Heba Abdelrasheed Allam, Enayat E. Aly, Ahmed K.B.A.W. Farouk, Ahmed M. El Kerdawy, Essam Rashwan, Safinaz E.S. Abbass. Design and Synthesis of some new 2,4,6-trisubstituted quinazoline EGFR inhibitors as targeted anticancer agents. Bioorganic Chemistry 2020; 98: 103726 doi: 10.1016/j.bioorg.2020.103726
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Vikas Pradhan, Salahuddin , Rajnish Kumar, Avijit Mazumder, Mohammad Mustaqeem Abdullah, Mohammad Shahar Yar, Mohamed Jawed Ahsan, Zabih Ullah. Molecular target interactions of quinoline derivatives as anticancer agents: A review. Chemical Biology & Drug Design 2023; 101(4): 977 doi: 10.1111/cbdd.14196
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Michaela Kuhlen, Jan-Henning Klusmann, Jessica I. Hoell. Molecular Approaches to Treating Pediatric Leukemias. Frontiers in Pediatrics 2019; 7 doi: 10.3389/fped.2019.00368
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Pascal Dao, Rafika Jarray, Nikaia Smith, Yves Lepelletier, Johanne Le Coq, Daniel Lietha, Réda Hadj-Slimane, Jean-Philippe Herbeuval, Christiane Garbay, Françoise Raynaud, Huixiong Chen. Inhibition of both focal adhesion kinase and fibroblast growth factor receptor 2 pathways induces anti-tumor and anti-angiogenic activities. Cancer Letters 2014; 348(1-2): 88 doi: 10.1016/j.canlet.2014.03.007
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Özge Sönmez, Nurgül Özgür Yurttaş, İlker İhtiyaroğlu, Halil Mete Çakır, Zeynep Atlı, Tuğrul Elverdi, Ayşe Salihoğlu, Nurhan Seyahi, Muhlis Cem Ar, Şeniz Öngören, Zafer Başlar, Teoman Soysal, Ahmet Emre Eşkazan. Effect of Tyrosine Kinase Inhibitor Therapy on Estimated Glomerular Filtration Rate in Patients with Chronic Myeloid Leukemia. Clinical Lymphoma Myeloma and Leukemia 2024; 24(4): 232 doi: 10.1016/j.clml.2023.12.004
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Liling Huang, Shiyu Jiang, Yuankai Shi. Tyrosine kinase inhibitors for solid tumors in the past 20 years (2001–2020). Journal of Hematology & Oncology 2020; 13(1) doi: 10.1186/s13045-020-00977-0
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